Benzofurocain

Chemical name

Ethyl ester 5-гидрокси-6-диметилам��нометил-2-метил-4-хлор��ензофуран-3- carboxylic acid tartrat

Gross

C34-H40-N2-014

Characteristics

White with Navy blue or svetlo-kremovogo coloured crystalline powder odourless. Rat in the water, not soluble in alcohol.

Of drugs

Drugs, the pain, местноанестезирующее . Oppressing synthesis prostaglandines has antibradikininovmi properties. Provides central analgezirutee and mestnoanestezirutee effect. Do the okshibutirata sodium and fentanyl in urgent surgical interventions (especially in patients with reduced functional reserves organism).

Indications

Pain syndrome of different genesis : pancreatitis (acute, chronic, including recurrent), peritonitis, hepatic and / or renal kolica, ischemic heart disease (stenocardia, myocardial infarction), acute pleurisy, bovine diseases and injuries peripheral nervous system (koreskove pain in the face of osteochondrosis spine, nevralgia, rapid, etc.), artropatia exchange and inflammatory origin, malignant Novoobrazovania.v Dentistry : chronic pain, infiltrazionnaya anaesthesia, preventing inflammation and local oedema (pulpit, periodontit, opening fester, textile operations).

Contraindications

Hypersensitivity, swelling of the brain, brain haemorrhage, AV blockade (full or partial), liver and / or kidney failure.

Side-Effects

Dizziness, weakness, drowsiness; With the rapid on / in the introduction, chills, nausea, vomiting; In the m-a sensation at the injection.

Specific guidance

In order to enhance the impact of pain is recommended together with tranquilizers, spazmolitikami.

Patient interaction

Solution benzofurokaina compatible Solutions diazepam, fentanyl, droperidola, sodium Okshibutirata.vvidu acid pH should not be confused with the solution of an alkaline reaction (thiopental sodium gexenal etc.).

Precautions

The long term use (up to 2 months) in 1.5-2 weeks after the start of treatment should be to reduce the dose by 10 to 20%, due to the possibility of cumulation.

Dosing and Administration

V / m, / in (struino or drip) in the dose of 0.1-0.3 g (10-30 ml) 1-3 times a day with a maximum daily dose of 1 g (100 ml) .V / in struino : being slow (1 ml for 15), if necessary izotoniceski diluted solution of sodium chloride or 5% glucose solution in a ratio of 1:1 .V / in the drip : being slow (10-30 drops / min) in the dose of 10 mg / kg (up to 1 g), 1% solution diluted with the same solutions to 250-500 Ml.infiltratinaya anesthetic in dentistry : not lemons, being 2-5 ml of 1% solution in the area of a tooth, risk treatment. You can combine with a 0.1% solution of adrenaline.

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