Brilokain-adrenaline forte

Roman name

Brilocaine-adrenaline forte

The composition and the form of

1 glass cartridge from 1.8 ml solution for injection (Brilokain-adrenaline), ukuporenny on the one hand plunjeron and on the other hand a rubber plug, obkatanna aluminium cap with a rubber gasket, contains artikaina hydrochloride and gidrotartrata adrenaline (epinephrine) in the ratio of 1:200000; in a contour acheikova packing 10 pcs. , in a cardboard bundle 5 upakovok.1 glass cartridge from 1.8 ml solution for injection (Brilokain adrenaline-forte), ukuporenny on the one hand plunjeron and on the other hand a rubber plug, obkatanna aluminium cap with a rubber gasket, contains artikaina hydrochloride and gidrotartrata adrenaline (epinephrine) in the ratio of 1:100000; in a contour acheikova packing 10 pcs. , in a cardboard bundle five packages.

Of drugs

Mestnoanestezirutee, sossoudossouerveshchee.

Pharmacokinetics

Artikain binds to plasma proteins at a 95% metabolized in the liver, excreted kidneys (63% in 6900), T_1/2 -25 min. Penetrates through the placental barrier.

Farmakodinamika

The fast begins-after 1-3 minutes and lasts for 45 minutes.

Indications

Anaesthesia (infiltrazionnaya and provodnikova) in Dentistry at ekstirpace tooth and sealing cavity machining teeth under crown.

Pregnancy and lactation

Perhaps.

Contraindications

Hypersensitivity, paroxizmalnaya tachycardia, tahiaritmia, bronchial asthma, glaucoma zakratougolnaya, simultaneous selective beta-adrenoblokatorov, severe liver failure, porphyria, vnutrisosudistye injections, Ray, the simultaneous admission of MAO inhibitors or tricyclic antidepressants, central nervous system diseases, malignant disease.

Side-Effects

From the nervous system and sensory organs : headache; Potential human consciousness until his loss; Violations breathing until it stops; Apnoea and muscle tremor, convulsions; Rarely produced in the eyes, diplopia, passing Slepota.so the circulatory system and blood (blood, gemostaz) : rarely arterial gipotenzia, tachycardia, aetiology, oppression cardiovascular Deatelnosti.so the respiratory system : despnoe, Apdimi.so part of the intestine : nausea, Rvota.allergicakie reactions : rhinitis, hyperemia skin, itching, angioneuroticeski swelling, swelling and inflammation at the injection; rarely anaphylactic shock.

Specific guidance

Deleting Danbury lower jaw in the uncomplicated infiltrazionnaya anaesthesia works provodnikovogo pain.

Patient interaction

Hypertensive effect can be reinforced tricyclic antidepressants and MAO inhibitors. Nor should designate product in the face of treatment neselektivei бета-адреноблокатора��и because of the increased risk of gipertoniceski kriza and expressed bradikardii.

Overdosing

Symptoms : dizziness, dwigatelnoe anxiety, impaired Soznaniya.lechenie : a patient horizontal position, in / with the introduction of barbiturates (with muscle podergivaniah or Generalized convulsions), in / in cefuroxim balanced elektrolitnykh and plazmozameshchath solutions in / with the introduction of glucocorticoids, adrenaline (in the case of threatening vascular collapse and growing bradikardii) the supply of oxygen, artificial respiration, if necessary endotrahealnaya intubation with controlled ventilation light, the use of peripheral vazodilatatorov if the AD.

Precautions

To be injected into the area of inflammation. In patients with a deficit compounds can be used only for urgent reasons (there is the likelihood of rollover and sometimes strengthen the drug).

Dosing and Administration

When you neoslojnennom teeth upper jaw, 1.8 ml (westibulyarnoe depot) at the tooth, if necessary, an additional 1.8 ml; Nebnom in terms warp or 0.1 ml (nebnoe depot); Professor with cavities and teeth to the teeth crowns (except molarov lower jaw), 0.5-1.8 ml per tooth (westibularnaya injection). Using any medical procedure adults can enter up to seven artikaina mg per kilogram body weight. The anaesthesia during which an intervention is 30-45 minutes.

Storage conditions

r-r d / in. : In the dark place at a temperature of no higher than 25 ° C. Avoid freezing

Shelf life

r-r d / in. : 2 grams.

Directory → Neurotropic funds → Local anaesthetics → Brilokain-adrenaline forte