Baclofen

Chemical name

бета-(Аминометил)-4-хло рбензолпропановая acid

Gross

C10-H12-Cl-N-O2

Characteristics

White or almost white crystalline powder, almost odourless. It is soluble in water, very little in methanol and nerastvorim in chloroform.

Of drugs

The drugs-miorelaksirutee, analgezirutee. GABA stimulates B-retseptora (braking), o 5b13 ppressing and mono polisinapticalkie though the spinalnom level, which reduces muscular tension and obesbolivatemu effect. Rapidly absorbed in the digestive tract. Not biotransformiroetsa. Report the news.

Indications

MS (to minimize muscle spasticnosti), schizophrenia disorder and alcoholism.

Restrictions on the use of

Violation of the kidney's age (up to 12 years). Be wary appoint persons profession which requires more attention and speed of reaction. During treatment nursing mothers should suspend breastfeeding. Not recommended sharing with alcohol and drugs, oppressive central nervous system.

Contraindications

Disorders, epilepsy, Parkinson's disease, pregnancy.

Side-Effects

Drowsiness, dizziness, weakness, sputannosti consciousness, human gait, nausea, vomiting, constipation, urine retention.

Patient interaction

Do effect of deprimiruth CNS.

Dosing and Administration

Inside, at the time of delivery. Initial dose of 5 mg three times a day. The maximum daily dose of 75-mg. Remove baclofen should gradually.

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